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Effects of Acute and Repeated Treatment with the Biased Mu Opioid Receptor Agonist TRV130 (Oliceridine) on Measures of Antinociception, Gastrointestinal Function & Abuse Liability in Rodents

RATIONALE: TRV130 (oliceridine; N-[(3-methoxythiophen-2-yl)methyl]-2-[(9R)-9-pyridin-2-yl-6-oxaspiro[4.5]decan-9-yl]ethanamine) is a novel mu opioid receptor (MOR) agonist that preferentially activates G-protein vs. β-arrestin signaling pathways coupled to MORs. Prevailing evidence suggests that TRV...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Veröffentlicht in:J Psychopharmacol
Hauptverfasser: Altarifi, Ahmad A., David, Bethany, Muchhala, Karan H., Blough, Bruce E., Akbarali, Hamid, Negus, S. Stevens
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2017
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5646680/
https://ncbi.nlm.nih.gov/pubmed/28142305
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1177/0269881116689257
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