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Distinct Signaling Patterns of Allosteric Antagonism at the P2Y(1) Receptor

Traditionally, G protein–coupled receptor antagonists are classified as competitive or noncompetitive and surmountable or insurmountable based on functional antagonism. P2Y(1) receptor (P2Y(1)R) structures showed two antagonists binding to two spatially distinct sites: nucleotide MRS2500 (orthosteri...

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Vydáno v:Mol Pharmacol
Hlavní autoři: Gao, Zhan-Guo, Jacobson, Kenneth A.
Médium: Artigo
Jazyk:Inglês
Vydáno: The American Society for Pharmacology and Experimental Therapeutics 2017
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5635520/
https://ncbi.nlm.nih.gov/pubmed/28864555
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.117.109660
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