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Antibody format and drug release rate determine the therapeutic activity of non-internalizing antibody-drug conjugates

The development of antibody-drug conjugates (ADCs), a promising class of anti-cancer agents, has traditionally relied on the use of antibodies capable of selective internalization in tumor cells. We have recently shown that also non-internalizing antibodies, coupled to cytotoxic drugs by means of di...

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Publicado en:Mol Cancer Ther
Main Authors: Gébleux, Rémy, Wulhfard, Sarah, Casi, Giulio, Neri, Dario
Formato: Artigo
Idioma:Inglês
Publicado: 2015
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5606287/
https://ncbi.nlm.nih.gov/pubmed/26294742
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1535-7163.MCT-15-0480
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