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New carboxamide derivatives bearing benzenesulphonamide as a selective COX-II inhibitor: Design, synthesis and structure-activity relationship

Sixteen new carboxamide derivatives bearing substituted benzenesulphonamide moiety (7a-p) were synthesized by boric acid mediated amidation of appropriate benzenesulphonamide with 2-amino-4-picoline and tested for anti-inflammatory activity. One compound 7c showed more potent anti-inflammatory activ...

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Détails bibliographiques
Publié dans:PLoS One
Auteurs principaux: Ugwu, David Izuchukwu, Okoro, Uchechukwu Chris, Ahmad, Hilal
Format: Artigo
Langue:Inglês
Publié: Public Library of Science 2017
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5602572/
https://ncbi.nlm.nih.gov/pubmed/28922386
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0183807
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