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Identification of 4-phenylquinolin-2(1H)-one as a specific allosteric inhibitor of Akt

Akt plays a major role in tumorigenesis and the development of specific Akt inhibitors as effective cancer therapeutics has been challenging. Here, we report the identification of a highly specific allosteric inhibitor of Akt through a FRET-based high-throughput screening, and characterization of it...

תיאור מלא

שמור ב:
מידע ביבליוגרפי
הוצא לאור ב:Sci Rep
Main Authors: Huang, Bill X., Newcomer, Kenny, Kevala, Karl, Barnaeva, Elena, Zheng, Wei, Hu, Xin, Patnaik, Samarjit, Southall, Noel, Marugan, Juan, Ferrer, Marc, Kim, Hee-Yong
פורמט: Artigo
שפה:Inglês
יצא לאור: Nature Publishing Group UK 2017
נושאים:
גישה מקוונת:https://ncbi.nlm.nih.gov/pmc/articles/PMC5601486/
https://ncbi.nlm.nih.gov/pubmed/28916818
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-017-11870-1
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