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Synthesis and In Vitro and In Vivo Evaluation of [(3)H]LRRK2-IN-1 as a Novel Radioligand for LRRK2

PURPOSE: LRRK2 (leucine-rich repeat kinase 2) has recently been proven to be a promising drug target for Parkinson’s disease (PD) due to an apparent enhanced activity caused by mutations associated with familial PD. To date, there have been no reports in which a LRRK2 inhibitor has been radiolabeled...

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Publicado en:Mol Imaging Biol
Autores principales: Malik, Noeen, Gifford, Andrew N, Sandell, Johan, Tuchman, Daniel, Ding, Yu-Shin
Formato: Artigo
Lenguaje:Inglês
Publicado: 2017
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5597475/
https://ncbi.nlm.nih.gov/pubmed/28289968
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11307-017-1070-1
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