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Decoding the selectivity of eIF2α holophosphatases and PPP1R15A inhibitors

The reversible phosphorylation of proteins controls most cellular functions. Protein kinases have been popular drug targets, unlike phosphatases, which remain a drug discovery challenge. Guanabenz and Sephin1 are selective inhibitors of the phosphatase regulatory subunit PPP1R15A (R15A) that prolong...

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Bibliografiske detaljer
Udgivet i:Nat Struct Mol Biol
Main Authors: Carrara, Marta, Sigurdardottir, Anna, Bertolotti, Anne
Format: Artigo
Sprog:Inglês
Udgivet: 2017
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5591645/
https://ncbi.nlm.nih.gov/pubmed/28759048
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nsmb.3443
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