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Targeting steroid hormone receptors for ubiquitination and degradation in breast and prostate cancer

Proteolysis targeting chimeric molecules (Protacs) target proteins for destruction by exploiting the ubiquitin-dependent proteolytic system of eukaryotic cells.We designed two Protacs that contain the peptide ‘degron’ from hypoxia-inducible factor-1α, which binds to the Von –Hippel–Lindau (VHL) E3 u...

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Detalles Bibliográficos
Publicado en:Oncogene
Autores principales: Rodriguez-Gonzalez, A, Cyrus, K, Salcius, M, Kim, K, Crews, CM, Deshaies, RJ, Sakamoto, KM
Formato: Artigo
Lenguaje:Inglês
Publicado: 2008
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5573236/
https://ncbi.nlm.nih.gov/pubmed/18794799
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/onc.2008.320
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