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PPARα Activation Suppresses Cytochrome P450 Induction Potential in Mice Treated with Gemfibrozil

Gemfibrozil, a peroxisome proliferator-activated receptor α (PPARα) agonist, is widely used for hypertriglyceridemia and mixed hyperlipidemia. Drug-drug interaction of gemfibrozil and other PPARα agonists has been reported. But the role of PPARα in Cytochrome P450 (CYP) induction by fibrates is not...

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Dettagli Bibliografici
Pubblicato in:Basic Clin Pharmacol Toxicol
Autori principali: Shi, Cunzhong, Min, Luo, Yang, Julin, Dai, Manyun, Song, Danjun, Hua, Huiying, Xu, Gangming, Gonzalez, Frank J., Liu, Aiming
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5554081/
https://ncbi.nlm.nih.gov/pubmed/28374976
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bcpt.12794
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