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Transition Metal-Free C3 Arylation of Indoles with Aryl Halides

Herein, we report an unprecedented transition metal-free, coupling of indoles with aryl halides. The reaction is promoted by KOtBu and is regioselective for C3 over nitrogen. The use of degassed solvents devoid of oxygen is necessary for the success of the transformation. Preliminary studies implica...

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Publié dans:Angew Chem Int Ed Engl
Auteurs principaux: Chen, Ji, Wu, Jimmy
Format: Artigo
Langue:Inglês
Publié: 2017
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5543986/
https://ncbi.nlm.nih.gov/pubmed/28256786
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.201612311
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