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Inhibitory effects and mechanism of dihydroberberine on hERG channels expressed in HEK293 cells

The human ether-a-go-go-related gene (hERG) potassium channel conducts rapid delayed rectifier potassium currents (I(Kr)) and contributes to phase III cardiac action potential repolarization. Drugs inhibit hERG channels by binding to aromatic residues in hERG helixes. Berberine (BBR) has multiple ac...

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Библиографические подробности
Опубликовано в: :PLoS One
Главные авторы: Yu, Dahai, Lv, Lin, Fang, Li, Zhang, Bo, Wang, Junnan, Zhan, Ge, Zhao, Lei, Zhao, Xin, Li, Baoxin
Формат: Artigo
Язык:Inglês
Опубликовано: Public Library of Science 2017
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5538702/
https://ncbi.nlm.nih.gov/pubmed/28763460
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0181823
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