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Associations of Drug Lipophilicity and Extent of Metabolism with Drug-Induced Liver Injury

Drug-induced liver injury (DILI), although rare, is a frequent cause of adverse drug reactions resulting in warnings and withdrawals of numerous medications. Despite the research community’s best efforts, current testing strategies aimed at identifying hepatotoxic drugs prior to human trials are not...

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Detalhes bibliográficos
Publicado no:Int J Mol Sci
Main Authors: McEuen, Kristin, Borlak, Jürgen, Tong, Weida, Chen, Minjun
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5535828/
https://ncbi.nlm.nih.gov/pubmed/28640208
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms18071335
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