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Steroidogenic metabolism of galeterone reveals a diversity of biochemical activities

Galeterone is a steroidal CYP17A1 inhibitor, androgen receptor (AR) antagonist and AR degrader, and was under evaluation in a phase III clinical trial for castration-resistant prostate cancer (CRPC). The A/B steroid ring (Δ(5), 3β-hydroxyl) structure of galeterone is identical to cholesterol, which...

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Detalhes bibliográficos
Publicado no:Cell Chem Biol
Main Authors: Alyamani, Mohammad, Li, Zhenfei, Berk, Michael, Li, Jianneng, Tang, Jingjie, Upadhyay, Sunil, Auchus, Richard J., Sharifi, Nima
Formato: Artigo
Idioma:Inglês
Publicado em: 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5533090/
https://ncbi.nlm.nih.gov/pubmed/28648378
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2017.05.020
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