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Tandem C(sp(3))–H Arylation/Oxidation and Arylation/Allylic Substitution of Isoindolinones

Isoindolinones comprise an important class of medicinally active compounds. Herein we report a straightforward functionalization of the isoindolinones with aryl bromides (22 examples) using a Pd(OAc)(2)/NIXANTPHOS-based catalyst system. Additionally 3-aryl 3-hydroxy isoindolinone derivatives, which...

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Dettagli Bibliografici
Pubblicato in:Adv Synth Catal
Autori principali: Jiménez, Jacqueline, Kim, Byeong-Seon, Walsh, Patrick J.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5482541/
https://ncbi.nlm.nih.gov/pubmed/28652858
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/adsc.201600654
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