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TRTH-33. COMPARATIVE PLASMA AND CEREBROSPINAL FLUID PHARMACOKINETICS OF BRAF AND MEK INHIBITORS IN A NONHUMAN PRIMATE MODEL

PURPOSE: BRAF(V600E) mutations are present in several pediatric CNS tumors, particularly pilocytic astrocytomas, gangliogliomas and pleomorphic xanthochromic astrocytomas. Several BRAF inhibitors are under clinical investigation, alone and in combination with MEK inhibitors. To guide the clinical de...

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Опубликовано в: :Neuro Oncol
Главные авторы: Rodgers, Louis, M Lester McCully, Cynthia, Gross, Andrea, Peer, Cody, Cruz, Rafael, Figg, William D, Widemann, Brigette, Warren, Katherine
Формат: Artigo
Язык:Inglês
Опубликовано: Oxford University Press 2017
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5475218/
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/neuonc/nox083.243
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