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Long-range allosteric regulation of the human 26S proteasome by 20S proteasome-targeting cancer drugs

The proteasome holoenzyme is the major non-lysosomal protease; its proteolytic activity is essential for cellular homeostasis. Thus, it is an attractive target for the development of chemotherapeutics. While the structural basis of core particle (CP) inhibitors is largely understood, their structura...

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Bibliografiska uppgifter
I publikationen:Nat Commun
Huvudupphovsmän: Haselbach, David, Schrader, Jil, Lambrecht, Felix, Henneberg, Fabian, Chari, Ashwin, Stark, Holger
Materialtyp: Artigo
Språk:Inglês
Publicerad: Nature Publishing Group 2017
Ämnen:
Länkar:https://ncbi.nlm.nih.gov/pmc/articles/PMC5458511/
https://ncbi.nlm.nih.gov/pubmed/28541292
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/ncomms15578
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