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Chemical probes targeting epigenetic proteins: Applications beyond oncology

Epigenetic chemical probes are potent, cell-active, small molecule inhibitors or antagonists of specific domains in a protein; they have been indispensable for studying bromodomains and protein methyltransferases. The Structural Genomics Consortium (SGC), comprising scientists from academic and phar...

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Detalhes bibliográficos
Publicado no:Epigenetics
Main Authors: Ackloo, Suzanne, Brown, Peter J., Müller, Susanne
Formato: Artigo
Idioma:Inglês
Publicado em: Taylor & Francis 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5453191/
https://ncbi.nlm.nih.gov/pubmed/28080202
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/15592294.2017.1279371
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