Cargando...

Targeted radionuclide therapy with astatine-211: Oxidative dehalogenation of astatobenzoate conjugates

(211)At is a most promising radionuclide for targeted alpha therapy. However, its limited availability and poorly known basic chemistry hamper its use. Based on the analogy with iodine, labelling is performed via astatobenzoate conjugates, but in vivo deastatination occurs, particularly when the con...

Descrición completa

Gardado en:
Detalles Bibliográficos
Publicado en:Sci Rep
Main Authors: Teze, David, Sergentu, Dumitru-Claudiu, Kalichuk, Valentina, Barbet, Jacques, Deniaud, David, Galland, Nicolas, Maurice, Rémi, Montavon, Gilles
Formato: Artigo
Idioma:Inglês
Publicado: Nature Publishing Group UK 2017
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5451414/
https://ncbi.nlm.nih.gov/pubmed/28566709
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-017-02614-2
Tags: Engadir etiqueta
Sen Etiquetas, Sexa o primeiro en etiquetar este rexistro!