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Identification and characterization of PKF118-310 as a KDM4A inhibitor

Epigenetic modifications are functionally involved in gene expression regulation. In particular, histone posttranslational modifications play a crucial role in functional chromatin organization. Several drugs able to inhibit or stimulate some families of proteins involved in epigenetic histone regul...

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Detalles Bibliográficos
Publicado en:Epigenetics
Main Authors: Franci, Gianluigi, Sarno, Federica, Nebbioso, Angela, Altucci, Lucia
Formato: Artigo
Idioma:Inglês
Publicado: Taylor & Francis 2016
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5406213/
https://ncbi.nlm.nih.gov/pubmed/27767379
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/15592294.2016.1249089
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