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Conformational dynamics of cathepsin D and binding to a small-molecule BACE1 inhibitor

BACE1 is a major therapeutic target for prevention and treatment of Alzheimer’s disease. Developing inhibitors that can selectively target BACE1 in favor of other proteases, especially cathepsin D (CatD), has presented significant challenges. Here we investigate the conformational dynamics and proto...

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Bibliographische Detailangaben
Veröffentlicht in:J Comput Chem
Hauptverfasser: Ellis, Christopher R., Tsai, Cheng-Chieh, Lin, Fang-Yu, Shen, Jana
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2017
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5403572/
https://ncbi.nlm.nih.gov/pubmed/28370344
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/jcc.24719
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