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Effect of Disease-Related Changes in Plasma Albumin on the Pharmacokinetics of Naproxen in Male and Female Arthritic Rats

Naproxen (NPX) is used in the treatment of rheumatoid arthritis (RA) for alleviation of pain and inflammation. In view of the extensive albumin binding of NPX, this study investigates whether chronic inflammation and sex influence the physiologic albumin concentrations, plasma protein binding, and p...

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Dades bibliogràfiques
Publicat a:Drug Metab Dispos
Autors principals: Li, Xiaonan, DuBois, Debra C., Almon, Richard R., Jusko, William J.
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2017
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5399645/
https://ncbi.nlm.nih.gov/pubmed/28246126
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.116.074500
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