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Design and Development of Fluorescent Vemurafenib Analogs for In Vivo Imaging

Herein we describe fluorescent derivatives of vemurafenib to probe therapeutic BRAF inhibition in live cells and in vivo. The compounds were evaluated and compared by determining target binding, inhibition of mutant BRAF melanoma cell lines and live cell imaging. We show that vemurafenib-BODIPY is a...

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發表在:Theranostics
Main Authors: Mikula, Hannes, Stapleton, Shawn, Kohler, Rainer H., Vinegoni, Claudio, Weissleder, Ralph
格式: Artigo
語言:Inglês
出版: Ivyspring International Publisher 2017
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在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC5399591/
https://ncbi.nlm.nih.gov/pubmed/28435463
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.7150/thno.18238
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