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Design and Development of Fluorescent Vemurafenib Analogs for In Vivo Imaging

Herein we describe fluorescent derivatives of vemurafenib to probe therapeutic BRAF inhibition in live cells and in vivo. The compounds were evaluated and compared by determining target binding, inhibition of mutant BRAF melanoma cell lines and live cell imaging. We show that vemurafenib-BODIPY is a...

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Dettagli Bibliografici
Pubblicato in:Theranostics
Autori principali: Mikula, Hannes, Stapleton, Shawn, Kohler, Rainer H., Vinegoni, Claudio, Weissleder, Ralph
Natura: Artigo
Lingua:Inglês
Pubblicazione: Ivyspring International Publisher 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5399591/
https://ncbi.nlm.nih.gov/pubmed/28435463
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.7150/thno.18238
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