Nalaganje...

Design and Development of Fluorescent Vemurafenib Analogs for In Vivo Imaging

Herein we describe fluorescent derivatives of vemurafenib to probe therapeutic BRAF inhibition in live cells and in vivo. The compounds were evaluated and compared by determining target binding, inhibition of mutant BRAF melanoma cell lines and live cell imaging. We show that vemurafenib-BODIPY is a...

Popoln opis

Shranjeno v:
Bibliografske podrobnosti
izdano v:Theranostics
Main Authors: Mikula, Hannes, Stapleton, Shawn, Kohler, Rainer H., Vinegoni, Claudio, Weissleder, Ralph
Format: Artigo
Jezik:Inglês
Izdano: Ivyspring International Publisher 2017
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC5399591/
https://ncbi.nlm.nih.gov/pubmed/28435463
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.7150/thno.18238
Oznake: Označite
Brez oznak, prvi označite!