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Increasing Thyromimetic Potency Through Halogen Substitution

Sobetirome is one of the most studied TRβ-selective thyromimetics in the field due to its excellent selectivity and potency. A small structural change - replacing the 3,5-dimethyl groups of sobetirome with either chlorine or bromine - produces significantly more potent compounds, both in vitro and i...

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Publicado en:ChemMedChem
Main Authors: Devereaux, Jordan, Ferrara, Skylar J., Banerji, Tania, Placzek, Andrew, Scanlan, Thomas S.
Formato: Artigo
Idioma:Inglês
Publicado: 2016
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5389920/
https://ncbi.nlm.nih.gov/pubmed/27731931
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.201600408
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