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A structure- and chemical genomics-based approach for repositioning of drugs against VCP/p97 ATPase

Valosin-containing protein (VCP/p97) ATPase (a.k.a. Cdc48) is a key member of the ER-associated protein degradation (ERAD) pathway. ERAD and VCP/p97 have been implicated in a multitude of human diseases, such as neurodegenerative diseases and cancer. Inhibition of VCP/p97 induces proteotoxic ER stre...

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Detalhes bibliográficos
Publicado no:Sci Rep
Main Authors: Segura-Cabrera, Aldo, Tripathi, Reshmi, Zhang, Xiaoyi, Gui, Lin, Chou, Tsui-Fen, Komurov, Kakajan
Formato: Artigo
Idioma:Inglês
Publicado em: Nature Publishing Group 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5359624/
https://ncbi.nlm.nih.gov/pubmed/28322292
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep44912
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