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Structural Requirements of HDAC Inhibitors: SAHA Analogues Modified at the C2 Position Display HDAC6/8 Selectivity

[Image: see text] Histone deacetylase (HDAC) proteins are epigenetic regulators that deacetylate protein substrates, leading to subsequent changes in cell function. HDAC proteins are implicated in cancers, and several HDAC inhibitors have been approved by the FDA as anticancer drugs, including SAHA...

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Bibliografiske detaljer
Udgivet i:ACS Med Chem Lett
Main Authors: Negmeldin, Ahmed T., Padige, Geetha, Bieliauskas, Anton V., Pflum, Mary Kay H.
Format: Artigo
Sprog:Inglês
Udgivet: American Chemical Society 2017
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5346987/
https://ncbi.nlm.nih.gov/pubmed/28337317
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.6b00124
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