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Cooperativity between Verapamil and ATP Bound to the Efflux Transporter P-glycoprotein

The P-glycoprotein (Pgp) transporter plays a central role in drug disposition by effluxing a chemically diverse range of drugs from cells through conformational changes and ATP hydrolysis. A number of drugs are known to activate ATP hydrolysis of Pgp, but coupling between ATP and drug binding is not...

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Publicado en:Biochem Pharmacol
Autores principales: Ledwitch, Kaitlyn V., Gibbs, Morgan E., Barnes, Robert W., Roberts, Arthur G.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2016
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5341695/
https://ncbi.nlm.nih.gov/pubmed/27531061
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2016.08.013
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