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PARP inhibitors: review of mechanisms of action and BRCA1/2 mutation targeting

Poly(ADP-ribose) polymerases have shown true promise in early clinical studies due to reported activity in BRCA-associated cancers. PARP inhibitors may represent a potentially important new class of chemotherapeutic agents directed at targeting cancers with defective DNA-damage repair. In order to w...

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Dettagli Bibliografici
Pubblicato in:Prz Menopauzalny
Autori principali: Dziadkowiec, Karolina N., Gąsiorowska, Emilia, Nowak-Markwitz, Ewa, Jankowska, Anna
Natura: Artigo
Lingua:Inglês
Pubblicazione: Termedia Publishing House 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5327624/
https://ncbi.nlm.nih.gov/pubmed/28250726
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.5114/pm.2016.65667
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