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Rapid and Reliable Binding Affinity Prediction of Bromodomain Inhibitors: A Computational Study

[Image: see text] Binding free energies of bromodomain inhibitors are calculated with recently formulated approaches, namely ESMACS (enhanced sampling of molecular dynamics with approximation of continuum solvent) and TIES (thermodynamic integration with enhanced sampling). A set of compounds is pro...

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Pubblicato in:J Chem Theory Comput
Autori principali: Wan, Shunzhou, Bhati, Agastya P., Zasada, Stefan J., Wall, Ian, Green, Darren, Bamborough, Paul, Coveney, Peter V.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Chemical Society 2016
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5312866/
https://ncbi.nlm.nih.gov/pubmed/28005370
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jctc.6b00794
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