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Drug trapping in hERG K(+) channels: (not) a matter of drug size?

Inhibition of hERG K(+) channels by structurally diverse drugs prolongs the ventricular action potential and increases the risk of torsade de pointes arrhythmias and sudden cardiac death. The capture of drugs behind closed channel gates, so-called drug trapping, is suggested to harbor an increased p...

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Shranjeno v:
Bibliografske podrobnosti
izdano v:Medchemcomm
Main Authors: Linder, Tobias, Bernsteiner, Harald, Saxena, Priyanka, Bauer, Florian, Erker, Thomas, Timin, Eugen, Hering, Steffen, Stary-Weinzinger, Anna
Format: Artigo
Jezik:Inglês
Izdano: Royal Society of Chemistry 2016
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC5292991/
https://ncbi.nlm.nih.gov/pubmed/28337337
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c5md00443h
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