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Drug trapping in hERG K(+) channels: (not) a matter of drug size?

Inhibition of hERG K(+) channels by structurally diverse drugs prolongs the ventricular action potential and increases the risk of torsade de pointes arrhythmias and sudden cardiac death. The capture of drugs behind closed channel gates, so-called drug trapping, is suggested to harbor an increased p...

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Dettagli Bibliografici
Pubblicato in:Medchemcomm
Autori principali: Linder, Tobias, Bernsteiner, Harald, Saxena, Priyanka, Bauer, Florian, Erker, Thomas, Timin, Eugen, Hering, Steffen, Stary-Weinzinger, Anna
Natura: Artigo
Lingua:Inglês
Pubblicazione: Royal Society of Chemistry 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5292991/
https://ncbi.nlm.nih.gov/pubmed/28337337
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c5md00443h
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