Wordt geladen...

Drug trapping in hERG K(+) channels: (not) a matter of drug size?

Inhibition of hERG K(+) channels by structurally diverse drugs prolongs the ventricular action potential and increases the risk of torsade de pointes arrhythmias and sudden cardiac death. The capture of drugs behind closed channel gates, so-called drug trapping, is suggested to harbor an increased p...

Volledige beschrijving

Bewaard in:
Bibliografische gegevens
Gepubliceerd in:Medchemcomm
Hoofdauteurs: Linder, Tobias, Bernsteiner, Harald, Saxena, Priyanka, Bauer, Florian, Erker, Thomas, Timin, Eugen, Hering, Steffen, Stary-Weinzinger, Anna
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: Royal Society of Chemistry 2016
Onderwerpen:
Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5292991/
https://ncbi.nlm.nih.gov/pubmed/28337337
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c5md00443h
Tags: Voeg label toe
Geen labels, Wees de eerste die dit record labelt!