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Metabolically labile fumarate esters impart kinetic selectivity to irreversible inhibitors

Electrophilic small molecules are an important class of chemical probes and drugs that produce biological effects by irreversibly modifying proteins. Examples of electrophilic drugs include covalent kinase inhibitors that are used to treat cancer and the multiple sclerosis drug dimethyl fumarate. Op...

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Detalhes bibliográficos
Publicado no:J Am Chem Soc
Main Authors: Zaro, Balyn W., Whitby, Landon R., Lum, Kenneth M., Cravatt, Benjamin F.
Formato: Artigo
Idioma:Inglês
Publicado em: 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5273863/
https://ncbi.nlm.nih.gov/pubmed/27960302
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jacs.6b10589
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