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Tissue Penetration of a Novel Spectinamide Antibiotic for the Treatment of Tuberculosis

The in vivo biodistribution and pharmacokinetics of 1329, a novel spectinamide antibiotic with anti-tubercular activity, were studied during intravenous administration of an tritium-labeled compound for nine consecutive, 12-hourly doses to rats. Serial blood samples were collected after the first an...

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Dades bibliogràfiques
Publicat a:AAPS J
Autors principals: Madhura, Dora Babu, Trivedi, Ashit, Liu, Jiuyu, Boyd, Vincent A., Jeffries, Cynthia, Loveless, Vivian, Lee, Richard E., Meibohm, Bernd
Format: Artigo
Idioma:Inglês
Publicat: Springer US 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5256617/
https://ncbi.nlm.nih.gov/pubmed/26984832
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12248-016-9900-7
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