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Base mutation analysis of topoisomerase II-idarubicin-DNA ternary complex formation. Evidence for enzyme subunit cooperativity in DNA cleavage.

Antitumor drugs, such as anthracyclines, interfere with mammalian DNA topoisomerase II by forming a ternary complex, DNA-drug-enzyme, in which DNA strands are cleaved and covalently linked to the enzyme. In this work, a synthetic 36-bp DNA oligomer derived from SV40 and mutated variants were used to...

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Detaylı Bibliyografya
Asıl Yazarlar: Bigioni, M, Zunino, F, Capranico, G
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: 1994
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC523684/
https://ncbi.nlm.nih.gov/pubmed/8036155
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