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Small molecule inhibitors of histone acetyltransferases and deacetylases are potential drugs for inflammatory diseases

Lysine acetylation is a reversible post-translational modification (PTM) of cellular proteins and represents an important regulatory switch in signal transduction. Lysine acetylation, in combination with other PTMs, directs the outcomes as well as the activation levels of important signal transducti...

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Pubblicato in:Drug Discov Today
Autori principali: Dekker, Frank J., van den Bosch, Thea, Martin, Nathaniel I.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2011
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5218544/
https://ncbi.nlm.nih.gov/pubmed/21477662
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.drudis.2011.03.009
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