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A four-compartment PBPK heart model accounting for cardiac metabolism - model development and application

In the field of cardiac drug efficacy and safety assessment, information on drug concentration in heart tissue is desirable. Because measuring drug concentrations in human cardiac tissue is challenging in healthy volunteers, mathematical models are used to cope with such limitations. With a goal of...

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Enregistré dans:
Détails bibliographiques
Publié dans:Sci Rep
Auteurs principaux: Tylutki, Zofia, Polak, Sebastian
Format: Artigo
Langue:Inglês
Publié: Nature Publishing Group 2017
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5209692/
https://ncbi.nlm.nih.gov/pubmed/28051093
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep39494
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