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Potent Inhibitors of Acetyltransferase Eis Overcome Kanamycin Resistance in Mycobacterium tuberculosis

A major cause of tuberculosis (TB) resistance to the aminoglycoside kanamycin (KAN) is the Mycobacterium tuberculosis (Mtb) acetyltransferase Eis. Upregulation of this enzyme is responsible for inactivation of KAN through acetylation of its amino groups. A 123 000-compound high-throughput screen (HT...

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Dettagli Bibliografici
Pubblicato in:ACS Chem Biol
Autori principali: Willby, Melisa J., Green, Keith D., Gajadeera, Chathurada S., Hou, Caixia, Tsodikov, Oleg V., Posey, James E., Garneau-Tsodikova, Sylvie
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5150266/
https://ncbi.nlm.nih.gov/pubmed/27010218
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.6b00110
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