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Synthesis of Triphenylethylene Bisphenols as Aromatase Inhibitors that Also Modulate Estrogen Receptors

A series of triphenylethylene bisphenol analogues of the selective estrogen receptor modulator (SERM) tamoxifen were synthesized and evaluated for their abilities to inhibit aromatase, bind to estrogen receptor-α (ER-α) and estrogen receptor-β (ER-β), and antagonize the activity of β-estradiol in MC...

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Dades bibliogràfiques
Publicat a:J Med Chem
Autors principals: Lv, Wei, Liu, Jinzhong, Skaar, Todd C., O'Neill, Elizaveta, Yu, Ge, Flockhart, David A., Cushman, Mark
Format: Artigo
Idioma:Inglês
Publicat: 2015
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5126733/
https://ncbi.nlm.nih.gov/pubmed/26704594
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.5b01677
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