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Development and validation of a novel LC–MS/MS method for simultaneous determination of abiraterone and its seven steroidal metabolites in human serum: Innovation in separation of diastereoisomers without use of a chiral column

Abiraterone acetate (AA), the prodrug of abiraterone, is FDA-approved for the treatment of castration-resistant prostate cancer. Abiraterone is metabolized in patients to a more potent analogue, D4A. However, we have recently reported that this analogue is further metabolized to additional metabolit...

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Detalles Bibliográficos
Publicado en:J Steroid Biochem Mol Biol
Autores principales: Alyamani, Mohammad, Li, Zhenfei, Upadhyay, Sunil K., Anderson, David J., Auchus, Richard J., Sharifi, Nima
Formato: Artigo
Lenguaje:Inglês
Publicado: 2016
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5124534/
https://ncbi.nlm.nih.gov/pubmed/27063554
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.jsbmb.2016.04.002
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