Loading...

Chemically Linked Vemurafenib Inhibitors Promote an Inactive BRAF(V600E) Conformation

The BRAF kinase, within the mitogen activated protein kinase (MAPK) signaling pathway, harbors activating mutations in about half of melanomas and to a significant extent in many other cancers. A single valine to glutamic acid substitution at residue 600 (BRAF(V600E)) accounts for about 90% of these...

Fuld beskrivelse

Na minha lista:
Bibliografiske detaljer
Udgivet i:ACS Chem Biol
Main Authors: Grasso, Michael, Estrada, Michelle A., Ventocilla, Christian, Samanta, Minu, Maksimoska, Jasna, Villanueva, Jessie, Winkler, Jeffrey D., Marmorstein, Ronen
Format: Artigo
Sprog:Inglês
Udgivet: 2016
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5108658/
https://ncbi.nlm.nih.gov/pubmed/27571413
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.6b00529
Tags: Tilføj Tag
Ingen Tags, Vær først til at tagge denne postø!