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Histone deacetylase inhibitors for cancer therapy: An evolutionarily ancient resistance response may explain their limited success

Histone deacetylase inhibitors (HDACi) are in clinical trials against a variety of cancers. Despite early successes, results against the more common solid tumors have been mixed. How is it that so many cancers, and most normal cells, tolerate the disruption caused by HDACi‐induced protein hyperacety...

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Publicat a:Bioessays
Autors principals: Halsall, John A., Turner, Bryan M.
Format: Artigo
Idioma:Inglês
Publicat: John Wiley and Sons Inc. 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5091640/
https://ncbi.nlm.nih.gov/pubmed/27717012
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/bies.201600070
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