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Inulanolide A as a new dual inhibitor of NFAT1-MDM2 pathway for breast cancer therapy

The transcription factor NFAT1 and the oncogene MDM2 have crucial roles in breast cancer development, progression, and metastasis. We have recently discovered that NFAT1 activates MDM2 expression. Here, we identified a small molecule (named Inulanolide A) that dually inhibited both NFAT1 and MDM2 in...

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Опубликовано в: :Oncotarget
Главные авторы: Qin, Jiang-Jiang, Wang, Wei, Sarkar, Sushanta, Voruganti, Sukesh, Agarwal, Rajesh, Zhang, Ruiwen
Формат: Artigo
Язык:Inglês
Опубликовано: Impact Journals LLC 2016
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5078034/
https://ncbi.nlm.nih.gov/pubmed/27105525
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.18632/oncotarget.8873
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