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Macrocycle-Based Hydroxamate Ligands for Complexation and Immunoconjugation of (89)Zirconium for Positron Emission Tomography (PET) Imaging

Four novel chelators (L1–L4) and their (89)zirconium complexes were prepared and compared with the (89)zirconium desferrioxamine B (DFO) complex. The new chelates are based on 1,4,7,10-tetraazacyclododecane (cyclen) and 1,4,8,11-tetraazacyclotetradecane (cyclam) scaffolds and present either three or...

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Publicado en:Chempluschem
Autores principales: Boros, Eszter, Holland, Jason P., Kenton, Nathaniel, Rotile, Nicholas, Caravan, Peter
Formato: Artigo
Lenguaje:Inglês
Publicado: 2016
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5019580/
https://ncbi.nlm.nih.gov/pubmed/27630807
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cplu.201600003
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