Učitavanje...

Mutation of Gly(721) Alters DNA Topoisomerase I Active Site Architecture and Sensitivity to Camptothecin

DNA topoisomerase I (Top1p) catalyzes the relaxation of supercoiled DNA via a concerted mechanism of DNA strand cleavage and religation. Top1p is the cellular target of the anticancer drug camptothecin (CPT), which reversibly stabilizes a covalent enzyme-DNA intermediate. Top1p clamps around duplex...

Cijeli opis

Spremljeno u:
Bibliografski detalji
Izdano u:J Biol Chem
Glavni autori: van der Merwe, Marie, Bjornsti, Mary-Ann
Format: Artigo
Jezik:Inglês
Izdano: 2007
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4995888/
https://ncbi.nlm.nih.gov/pubmed/18056711
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M705781200
Oznake: Dodaj oznaku
Bez oznaka, Budi prvi tko označuje ovaj zapis!