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Molecular Basis for Redox Activation of Epidermal Growth Factor Receptor Kinase

EGFR is a target of signal-derived H(2)O(2) and oxidation of active site cysteine 797 to sulfenic acid enhances kinase activity. Although a major class of covalent drugs targets C797, nothing is known about its catalytic importance or how S-sulfenylation leads to activation. Here, we report the firs...

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Dettagli Bibliografici
Pubblicato in:Cell Chem Biol
Autori principali: Truong, Thu H., Ung, Peter Man-Un, Palde, Prakash B., Paulsen, Candice E., Schlessinger, Avner, Carroll, Kate S.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4958504/
https://ncbi.nlm.nih.gov/pubmed/27427230
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2016.05.017
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