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Comparative Metabolism of Batracylin (NSC 320846) and N-acetylbatracylin (NSC 611001) Using Human, Dog, and Rat Preparations In Vitro

BACKGROUND: Batracylin is a heterocyclic arylamine topoisomerase inhibitor with preclinical anticancer activity. Marked species differences in sensitivity to the toxicity of batracylin were observed and attributed to differential formation of N-acetylbatracylin by N-acetyltransferase. A Phase I tria...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Veröffentlicht in:J Drug Metab Toxicol
Hauptverfasser: Covey, Joseph M, Reid, Joel M, Buhrow, Sarah A, Kuffel, Mary, Walden, Chad, Behrsing, Holger, Ames, Matthew M
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2016
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4948755/
https://ncbi.nlm.nih.gov/pubmed/27441096
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.4172/2157-7609.1000203
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