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MET Exon 14 Alterations in Lung Cancer: Exon Skipping Extends Half-Life

MET exon 14 alterations are a diverse group of mutations, many of which disrupt splice acceptor or donor sites leading to exon 14 skipping, impaired receptor degradation, and oncogenic transformation. These alterations are clinically targetable with MET-directed therapy.

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Detalles Bibliográficos
Publicado en:Clin Cancer Res
Autor principal: Drilon, Alexander
Formato: Artigo
Lenguaje:Inglês
Publicado: 2016
Materias:
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC4911276/
https://ncbi.nlm.nih.gov/pubmed/27009743
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1078-0432.CCR-16-0229
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