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Liposomal-mediated delivery of the p21 activated kinase-1 (PAK-1) inhibitorIPA-3limits prostate tumor growth in vivo

P21 activated kinases-1 (PAK-1)is implicated in various diseases. It is inhibited by thesmall molecule ‘Inhibitor targeting PAK1 activation-3’ (IPA-3), which is highly specific but metabolically unstable. To address this limitation we encapsulatedIPA-3 in sterically stabilized liposomes (SSL). SSL-I...

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Publicado en:Nanomedicine
Main Authors: Al-Azayzih, Ahmad, Missaoui, Wided N., Cummings, Brian S., Somanath, Payaningal R.
Formato: Artigo
Idioma:Inglês
Publicado: 2016
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4889517/
https://ncbi.nlm.nih.gov/pubmed/26949163
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.nano.2016.01.003
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