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Docking Screens for Novel Ligands Conferring New Biology

It is now plausible to dock libraries of 10 million molecules against targets over several days or weeks. When the molecules screened are commercially available, they may be rapidly tested to find new leads. Although docking retains important liabilities (it cannot calculate affinities accurately no...

Deskribapen osoa

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Xehetasun bibliografikoak
Argitaratua izan da:J Med Chem
Egile Nagusiak: Irwin, John J., Shoichet, Brian K.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2016
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC4865415/
https://ncbi.nlm.nih.gov/pubmed/26913380
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.5b02008
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