載入...

Synthesis of novel amide and urea derivatives of thiazol-2-ethylamines and their activity against Trypanosoma brucei rhodesiense

2-(2-Benzamido)ethyl-4-phenylthiazole (1) was one of 1035 molecules (grouped into 115 distinct scaffolds) found to be inhibitory to Trypanosoma brucei, the pathogen causing human African trypanosomiasis, at concentrations below 3.6 μM and non-toxic to mammalian (Huh7) cells in a phenotypic high-thro...

全面介紹

Na minha lista:
書目詳細資料
發表在:Bioorg Med Chem
Main Authors: Patrick, Donald A., Wenzler, Tanja, Yang, Sihyung, Weiser, Patrick T., Wang, Michael Zhuo, Brun, Reto, Tidwell, Richard R.
格式: Artigo
語言:Inglês
出版: 2016
主題:
在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC4862372/
https://ncbi.nlm.nih.gov/pubmed/27102161
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2016.04.006
標簽: 添加標簽
沒有標簽, 成為第一個標記此記錄!